Compile Data Set for Download or QSAR
Found 918 of ic50 data for polymerid = 50001330,50001957
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271230(US10059720, Example 45 | US10975091, Example 45)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271230(US10059720, Example 45 | US10975091, Example 45)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM284944(US10023583, Example 16)copy SMILEScopy InChI
Affinity DataIC50: 0.560nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29Z96X2US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM401319(US10005762, Example 3)copy SMILEScopy InChI
Affinity DataIC50: 0.580nMAssay Description:The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1V3QUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271290(US10059720, Example 105 | US10975091, Example 105)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271290(US10059720, Example 105 | US10975091, Example 105)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM401367(US10005762, Example 47)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1V3QUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271330(US10059720, Example 145 | US10975091, Example 145)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271257(US10059720, Example 72 | US10975091, Example 72)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271257(US10059720, Example 72 | US10975091, Example 72)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271330(US10059720, Example 145 | US10975091, Example 145)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM284942(US10023583, Example 14)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29Z96X2US Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271230(US10059720, Example 45 | US10975091, Example 45)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271230(US10059720, Example 45 | US10975091, Example 45)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271310(US10059720, Example 125 | US10975091, Example 125)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271310(US10059720, Example 125 | US10975091, Example 125)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271316(US10059720, Example 131 | US10975091, Example 131)copy SMILEScopy InChI
Affinity DataIC50: 0.910nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271316(US10059720, Example 131 | US10975091, Example 131)copy SMILEScopy InChI
Affinity DataIC50: 0.910nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271309(US10059720, Example 124 | US10975091, Example 124)copy SMILEScopy InChI
Affinity DataIC50: 0.920nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271309(US10059720, Example 124 | US10975091, Example 124)copy SMILEScopy InChI
Affinity DataIC50: 0.920nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271257(US10059720, Example 72 | US10975091, Example 72)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271257(US10059720, Example 72 | US10975091, Example 72)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM401355(US10005762, Example 35)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1V3QUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271275(US10059720, Example 90 | US10975091, Example 90)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271275(US10059720, Example 90 | US10975091, Example 90)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271318(US10059720, Example 133 | US10975091, Example 133)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271275(US10059720, Example 90 | US10975091, Example 90)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271275(US10059720, Example 90 | US10975091, Example 90)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271288(US10059720, Example 103 | US10975091, Example 103)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271198(US10059720, Example 13 | US10975091, Example 13)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271288(US10059720, Example 103 | US10975091, Example 103)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271198(US10059720, Example 13 | US10975091, Example 13)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271318(US10059720, Example 133 | US10975091, Example 133)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271277(US10059720, Example 92 | US10975091, Example 92)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271258(US10059720, Example 73 | US10975091, Example 73)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM284929(US10023583, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29Z96X2US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271277(US10059720, Example 92 | US10975091, Example 92)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271258(US10059720, Example 73 | US10975091, Example 73)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271190(US10059720, Example 6 | US10975091, Example 6)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271190(US10059720, Example 6 | US10975091, Example 6)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271213(US10059720, Example 28 | US10975091, Example 28)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271277(US10059720, Example 92 | US10975091, Example 92)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM401322(US10005762, Example 4(3))copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1V3QUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271213(US10059720, Example 28 | US10975091, Example 28)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271277(US10059720, Example 92 | US10975091, Example 92)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271260(US10059720, Example 75 | US10975091, Example 75)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271260(US10059720, Example 75 | US10975091, Example 75)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271243(US10059720, Example 58 | US10975091, Example 58)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271272(US10059720, Example 87 | US10975091, Example 87)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271198(US10059720, Example 13 | US10975091, Example 13)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
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